Protein Details: Potassium voltage-gated channel subfamily KQT member 3

Protein ID

ICDB_Pro_0640

Protein Name

Potassium voltage-gated channel subfamily KQT member 3

Gene Name

KCNQ3

Organism

Bos taurus (Bovine)

Length

866 amino acids

AlphaFoldDB

AF-P58126-F1-model_v4.pdb

Function

Associates with KCNQ2 or KCNQ5 to form a potassium channel with essentially identical properties to the channel underlying the native M-current; a slowly activating and deactivating potassium conductance which plays a critical role in determining the subthreshold electrical excitability of neurons as well as the responsiveness to synaptic inputs. Therefore; it is important in the regulation of neuronal excitability. KCNQ2-KCNQ3 channel is selectively permeable to other cations besides potassium; in decreasing order of affinity K(+) > Rb(+) > Cs(+) > Na(+). Associates with Na(+)-coupled myo-inositol symporter SLC5A3 forming a coregulatory complex that alters ion selectivity; increasing Na(+) and Cs(+) permeation relative to K(+) permeation

Sequence

MGLKARRPAGAAGGGGDGGGGGGGAANPAGGDAAAAGDEERKVGLAPGDVEQVTLALGAGADKDGTLLLEGGGRDEGQRRTPQGIGLLAKTPLSRPVKRNNAKYRRIQTLIYDALERPRGWALLYHALVFLIVLGCLILAVLTTFREYETVSGDWLLLLETFAIFIFGAEFALRIWAAGCCCRYKGWRGRLKFARKPLCMLDIFVLIASVPVVAVGNQGNVLATSLRSLRFLQILRMLRMDRRGGTWKLLGSAICAHSKELITAWYIGFLTLILSSFLVYLVEKDVPEVDAQGEEMKEEFETYADALWWGLITLATIGYGDKTPKTWEGRLIAATFSLIGVSFFALPAGILGSGLALKVQEQHRQKHFEKRRKPAAELIQAAWRYYATNPNRIDLVATWRFYESVVSFPFFRKEQLDPAASQKLGLLDRVRLSNPRGSNTKGKLFTPLNVDAIEESPSKEPKPVGSNNKERFRTAFRMKAYAFWQSSEDAGTGDPTAEDRGYGNDFLIEDMIPTLKAAIRAVRILQFRLYKKKFKETLRPYDVKDVIEQYSAGHLDMLSRIKYLQTRIDMIFTPGPPSTPKHKKSQRGAAFTYPSQQSPRNEPYVARPSTSETEDQSMMGKFVKVERQVHDMGKKLDFLVDMHLQHMERLQVHVAGFSPSKGASSPAEAEQKEDRRDADLKTIICNYSETGAPDAPYSFHQVPVDKVGPYGFFAHDPVNLPLGGPSSGKGHATPYAERPTVLPILTLLDSRGSYRSQVELHGPCSDRVSPRQRRSITRDSDTPLSLMSVNHEELERSPSGFSISQDRDDYAFGPSGGSSWMREKRYLAEGETDTDTEPFTPSGSLPLSSTGDGISDSIWTPSGKPT

PDB Structures

Ligand Binding

1. DICL_CP

2. DICL_Pep

Binding Site

Disease

Location

DOI ID

RefSeq

NP_776799.1

Feature